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酶学靶点筛选

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所在地: 湖北武汉市
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最后更新: 2018-08-20 13:40
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服务说明
 分子靶点筛选的药物发现途径越来越广泛的运用于新药的开发中,酶学研究在新药研发中的地位越来越重要。酶学实验涵盖600多种筛选模型,包括了常见的组蛋白去乙酰酶类,组蛋白去甲基化酶,酪氨酸激酶,丝氨酸激酶,甲基化转移酶,磷酸二酯酶,DNA修复酶,热休克蛋白,免疫相关蛋白等,以及激酶谱的筛选。
合研生物拥有丰富的酶学筛选经验,根据样本量的大小提供灵活的项目实施安排计划,可提供96孔和384孔两种板型的筛选模式,加速您的药物研发进程。

 

Cat#

Target

Assay

Format

Deacetylases

E001

HDAC

Fluorogenic assay

96 well

E002

HDAC1

Fluorogenic assay

96 well

E003

HDAC2

Fluorogenic assay

96 well

E004

HDAC3

Fluorogenic assay

96 well

E005

HDAC4

Fluorogenic assay

96 well

E006

HDAC5

Fluorogenic assay

96 well

E007

HDAC6

Fluorogenic assay

96 well

E008

HDAC7

Fluorogenic assay

96 well

E009

HDAC8

Fluorogenic assay

96 well

E010

HDAC9

Fluorogenic assay

96 well

E011

SIRT1

Fluorogenic assay

96 well

E012

SIRT2

Fluorogenic assay

96 well

E013

SIRT3

Fluorogenic assay

96 well

E014

SIRT5

Fluorogenic assay

96 well

Demethylases

E015

FBXL10

AlphaScreen assay/Chemiluminescent

96/384 well

E016

FBXL11

AlphaScreen assay

96/384 well

E017

JARID1A

AlphaScreen assay/Chemiluminescent

96/384 well

E018

JARID1B

AlphaScreen assay/Chemiluminescent

96/384 well

E019

JARID1C

AlphaScreen assay

96/384 well

E020

JHDM1D

AlphaScreen assay/Chemiluminescent

96/384 well

E021

JMJD1A

AlphaScreen assay

96/384 well

E022

LSD1

Fluorogenic assay

96/384 well

E023

JMJD2A

AlphaScreen assay

96/384 well

E024

JMJD2B

AlphaScreen assay

96/384 well

E025

JMJD2C

AlphaScreen assay/Chemiluminescent

96/384 well

E026

JMJD2D

Chemiluminescent assay

96/384 well

E027

JMJD2E

AlphaScreen assay

96/384 well

E028

JMJD3

AlphaScreen assay/Chemiluminescent

96/384 well

E029

PHF8

AlphaScreen assay

96/384 well

E030

TET1

Chemiluminescent assay

96 well

E031

TET2

Chemiluminescent assay

96 well

E032

UTX

AlphaScreen assay/Chemiluminescent

96/384 well

Methyltransferases

E033

DNMT

chemiluminescence

96 well

E034

DNMT1

chemiluminescence

96 well

E035

DNMT3A

chemiluminescence

96 well

E036

DNMT3B

chemiluminescence

96 well

E037

DOT1L

chemiluminescence

96 well

E038

EHMT1/GLP

chemiluminescence

96 well

E039

EZH1

chemiluminescence

96 well

E040

EZH2(A677G)

chemiluminescence

96 well

E041

EZH2(Y641F)

chemiluminescence

96 well

E042

EZH2(A641N)

chemiluminescence/TR-FRET

96 well

E043

G9a

chemiluminescence

96 well

E044

Histone H3(K9)

chemiluminescence

96 well

E045

Histone H4(R3)

AlphaScreen assay

96 well

E046

MLL1

chemiluminescence

96 well

E047

NSD1

chemiluminescence

96 well

E048

NSD2

chemiluminescence

96 well

E049

PRMT1

chemiluminescence/AlphaScreen assay

96 well

E050

PRMT3

chemiluminescence/AlphaScreen assay

96 well

E051

PRMT4

chemiluminescence

96 well

E052

PRMT5

chemiluminescence/TR-FRET

96/384 well

E053

PRMT8

chemiluminescence

96 well

E054

SETD2

chemiluminescence

96 well

E055

SetDB1

chemiluminescence

96 well

E056

SUV39H1

chemiluminescence

96 well

E057

SUV39H2

chemiluminescence

96 well

E058

SUV4-20H1

chemiluminescence

96 well

E059

EZH2(A378T)

chemiluminescence

96 well

E060

NSD3

chemiluminescence

96 well

E061

PRMT6

chemiluminescence/TR-FRET

96/384 well

E062

PRMT9

AlphaScreen assay

96 well

E063

SMYD2

chemiluminescence

96 well

E064

SMYD3

AlphaScreen assay

96 well

E065

SMYD4

chemiluminescence

96 well

E066

SET7/9

Fluorogenic assay

96 well

E067

SET8

Fluorogenic assay

96 well

Phosphodiesterase

E068

PDE

FP Assay

96 well

E069

PDE10A

TR-FRET

96 well

E070

PDE10A1

TR-FRET/ FP Assay

96 /384 well

E071

PDE10A2

FP Assay

96 well

E072

PDE11A

FP Assay

96 well

E073

PDE1A

FP Assay

96 well

E074

PDE1B

TR-FRET

96 well

E075

PDE1C

TR-FRET/ FP Assay

96 /384 well

E076

PDE2A

FP Assay/ FP Assay

96 /384 well

E077

PDE3A

TR-FRET

96 well

E078

PDE3B

FP Assay/ FP Assay

96 /384 well

E079

PDE4A

FP Assay

96 well

E080

PDE4B2

FP Assay

96 well

E081

PDE4D2

TR-FRET

96 well

E082

PDE4D3

TR-FRET

96 well

E083

PDE4D7

TR-FRET

96 well

E084

PDE5A1

FP Assay/ FP Assay

96 /384 well

E085

PDE7A

FP Assay/ FP Assay

96 /384 well

E086

PDE7B

FP Assay

96 well

E087

PDE8A

FP Assay

96 well

E088

PDE9A

FP Assay

96 well

E089

PDE4C

FP Assay

384 well

E090

Autotaxin

Fluorogenic assay

96 well

PARPs

E091

PARP1

chemiluminescence/Colorimetric Assay

96/384 well

E092

PARP2

chemiluminescence/Colorimetric Assay

96/384 well

E093

PARP3

chemiluminescence

96/384 well

E094

PARP6

chemiluminescence

96/384 well

E095

PARP7

chemiluminescence

96/384 well

E096

PARP10

chemiluminescence

96/384 well

E097

PARP11

chemiluminescence

96/384 well

E098

PARP14

chemiluminescence

96/384 well

E099

PARP15

chemiluminescence

96/384 well

E100

TNKS1

chemiluminescence

96/384 well

E101

TNKS2

chemiluminescence

96/384 well

Protease

E102

DPP3

Fluorogenic assay

96 well

E103

DPP4

Fluorogenic assay

96 well

E104

DPP7

Fluorogenic assay

96 well

E105

DPP8

Fluorogenic assay

96 well

E106

DPP9

Fluorogenic assay

96 well

E107

FAP

Fluorogenic assay

96 well

E108

POP

Fluorogenic assay

96 well

E109

Renin

Fluorogenic assay

96 well

E110

Caspase-3

Fluorogenic assay

96 well

E111

Caspase-6

Fluorogenic assay

96 well

E112

Caspase-7

Fluorogenic assay

96 well

E113

Caspase-8

Fluorogenic assay

96 well

Bromodomains

E114

ATAD2A

TR-FRET/AlphaScreen assay

96/384 well

E115

ATAD2B

TR-FRET/AlphaScreen assay

96/384 well

E116

BAZ2B

AlphaScreen assay

96/384 well

E117

BPTF/FALZ

TR-FRET

96/384 well

E118

BRD1

TR-FRET/AlphaScreen assay

96/384 well

E119

BRD2

TR-FRET/AlphaScreen assay

96/384 well

E120

BRD3

TR-FRET/AlphaScreen assay

96/384 well

E121

BRD4

TR-FRET/AlphaScreen assay

96/384 well

E122

BRD9

TR-FRET

96/384 well

E123

BRDT

TR-FRET

96/384 well

E124

BRPF3

TR-FRET/AlphaScreen assay

96/384 well

E125

CECR2

TR-FRET/AlphaScreen assay

96/384 well

E126

CREBBP

TR-FRET/AlphaScreen assay

96/384 well

E127

SMARCA2

TR-FRET/AlphaScreen assay

96/384 well

E128

SMARCA4

TR-FRET/AlphaScreen assay

96/384 well

E129

TAF1(BD2)

TR-FRET

96/384 well

E130

TAF1L(BD2)

TR-FRET

96/384 well

E131

TRIM24

TR-FRET

96/384 well

E132

WDR9/BRWD1

TR-FRET

96/384 well

E133

BACE1

TR-FRET

96/384 well

E134

BRG1

TR-FRET

96 well

E135

BRM

TR-FRET

96 well

E136

CBP

TR-FRET

96 well

Kinase

E137

ABL1

ADP-Glo

96/384 well

E138

ABL1(E255K)

ADP-Glo

96/384 well

E139

ABL1(T315I)

ADP-Glo

96/384 well

E140

ABL1(Y253F)

ADP-Glo

96/384 well

E141

ACK

ADP-Glo

96/384 well

E142

AKT1

ADP-Glo

96/384 well

E143

AKT2

ADP-Glo

96/384 well

E144

AKT3

ADP-Glo

96/384 well

E145

ALK2

ADP-Glo

96/384 well

E146

ALK4

ADP-Glo

96/384 well

E147

ALK6

ADP-Glo

96/384 well

E148

AMAPK(A1/B1/G2)

ADP-Glo

96/384 well

E149

AMPK(A1/B1/G1)

ADP-Glo

96/384 well

E150

AMPK(A2/B1/G1)

ADP-Glo

96/384 well

E151

ASK1

ADP-Glo

96/384 well

E152

Aurora A

ADP-Glo

96/384 well

E153

Aurora B

ADP-Glo

96/384 well

E154

AXL

ADP-Glo

96/384 well

E155

BRK

ADP-Glo

96/384 well

E156

BXM

ADP-Glo

96/384 well

E157

CAMK1γ

ADP-Glo

96/384 well

E158

CAMK2α

ADP-Glo

96/384 well

E159

CAMK2γ

ADP-Glo

96/384 well

E160

CAMKK1

ADP-Glo

96/384 well

E161

CDC7/DBF4

ADP-Glo

96/384 well

E162

CDK2/CyclinA2

ADP-Glo

96/384 well

E163

CDK2/CyclinE1

ADP-Glo

96/384 well

E164

CDK3/cyclinE1

ADP-Glo

96/384 well

E165

CDK5/p25

ADP-Glo

96/384 well

E166

CDK5/p35

ADP-Glo

96/384 well

E167

CDK6/CyclinD3

ADP-Glo

96/384 well

E168

CDK9/Cyclink

ADP-Glo

96/384 well

E169

CHK1

ADP-Glo

96/384 well

E170

CHK2

ADP-Glo

96/384 well

E171

CK1a1

ADP-Glo

96/384 well

E172

CK1γ1

ADP-Glo

96/384 well

E173

CK1ε

ADP-Glo

96/384 well

E174

CK2α1

ADP-Glo

96/384 well

E175

c-KIT

ADP-Glo

96/384 well

E176

CLK1

ADP-Glo

96/384 well

E177

CLK3

ADP-Glo

96/384 well

E178

c-MER

ADP-Glo

96/384 well

E179

CSK

ADP-Glo

96/384 well

E180

DAPK1

ADP-Glo

96/384 well

E181

DDR2

ADP-Glo

96/384 well

E182

DNA-PK

ADP-Glo

96/384 well

E183

DYRK2

ADP-Glo

96/384 well

E184

EGFR

ADP-Glo

96/384 well

E185

EGFR(L858R)

ADP-Glo

96/384 well

E186

EGFR(L861Q)

ADP-Glo

96/384 well

E187

EGFR(T790,L858R)

ADP-Glo

96/384 well

E188

EGFR(T790M)

ADP-Glo

96/384 well

E189

EIF2AK2

ADP-Glo

96/384 well

E190

EPHA1

ADP-Glo

96/384 well

E191

ERK1

ADP-Glo

96/384 well

E192

ERK2

ADP-Glo

96/384 well

E193

FAK

ADP-Glo

96/384 well

E194

FES

ADP-Glo

96/384 well

E195

FGFR1

ADP-Glo

96/384 well

E196

FGFR2

ADP-Glo

96/384 well

E197

FGFR3(K650E)

ADP-Glo

96/384 well

E198

FGFR4

ADP-Glo

96/384 well

E199

FLT1

ADP-Glo

96/384 well

E200

FLT3

ADP-Glo

96/384 well

E201

FLT3(D835Y)

ADP-Glo

96/384 well

E202

FMS

ADP-Glo

96/384 well

E203

FYN A

ADP-Glo

96/384 well

E204

GRK5

ADP-Glo

96/384 well

E205

GSK3α

ADP-Glo

96/384 well

E206

GSK3β

ADP-Glo

96/384 well

E207

HER2

ADP-Glo

96/384 well

E208

HER4

ADP-Glo

96/384 well

E209

HIPK1

ADP-Glo

96/384 well

E210

HPK1

ADP-Glo

96/384 well

E211

IGF1R

ADP-Glo

96/384 well

E212

IKK

ADP-Glo

96/384 well

E213

IKKα

ADP-Glo

96/384 well

E214

InsR

ADP-Glo

96/384 well

E215

IRAK4

ADP-Glo

96/384 well

E216

ITK

ADP-Glo

96/384 well

E217

JAK3

ADP-Glo

96/384 well

E218

JNK1

ADP-Glo

96/384 well

E219

JNK3

ADP-Glo

96/384 well

E220

KDR

ADP-Glo

96/384 well

E221

KHS1

ADP-Glo

96/384 well

E222

LCK

ADP-Glo

96/384 well

E223

Lipid kinase

ADP-Glo

96/384 well

E224

LRRK2

ADP-Glo

96/384 well

E225

LYN B

ADP-Glo

96/384 well

E226

MAPKAPK2

ADP-Glo

96/384 well

E227

MAPKAPK3

ADP-Glo

96/384 well

E228

MAPKAPK5

ADP-Glo

96/384 well

E229

MARK1

ADP-Glo

96/384 well

E230

MELK

ADP-Glo

96/384 well

E231

MET

ADP-Glo

96/384 well

E232

MET(M1250T)

ADP-Glo

96/384 well

E233

MINK1

ADP-Glo

96/384 well

E234

MLCK

ADP-Glo

96/384 well

E235

MLK1

ADP-Glo

96/384 well

E236

MLK2

ADP-Glo

96/384 well

E237

MRCKa

ADP-Glo

96/384 well

E238

MSK1

ADP-Glo

96/384 well

E239

MSK2

ADP-Glo

96/384 well

E240

MST1

ADP-Glo

96/384 well

E241

MYO3β

ADP-Glo

96/384 well

E242

Name

ADP-Glo

96/384 well

E243

NEK2

ADP-Glo

96/384 well

E244

NEK3

ADP-Glo

96/384 well

E245

NIK

ADP-Glo

96/384 well

E246

NUAK2

ADP-Glo

96/384 well

E247

p38α

ADP-Glo

96/384 well

E248

p38B

ADP-Glo

96/384 well

E249

p38γ

ADP-Glo

96/384 well

E250

P38δ

ADP-Glo

96/384 well

E251

p70S6K

ADP-Glo

96/384 well

E252

p70S6Kb

ADP-Glo

96/384 well

E253

PAK1/CDC42

ADP-Glo

96/384 well

E254

PAK3

ADP-Glo

96/384 well

E255

PAK4

ADP-Glo

96/384 well

E256

PASK

ADP-Glo

96/384 well

E257

PDGFRa(D842V)

ADP-Glo

96/384 well

E258

PDGFRa(T674I)

ADP-Glo

96/384 well

E259

PDGFRα

ADP-Glo

96/384 well

E260

PDGFRβ

ADP-Glo

96/384 well

E261

PDK1

ADP-Glo

96/384 well

E262

PI3K Lipid kinases

ADP-Glo

96/384 well

E263

PI3K-Glo

ADP-Glo

96/384 well

E264

PIM1

ADP-Glo

96/384 well

E265

PIM2

ADP-Glo

96/384 well

E266

PKA

ADP-Glo

96/384 well

E267

PKC

ADP-Glo

96/384 well

E268

PKC1

ADP-Glo

96/384 well

E269

PKCα

ADP-Glo

96/384 well

E270

PKCβII

ADP-Glo

96/384 well

E271

PKCγ

ADP-Glo

96/384 well

E272

PKCδ

ADP-Glo

96/384 well

E273

PKCε

ADP-Glo

96/384 well

E274

PKCζ

ADP-Glo

96/384 well

E275

PKCθ

ADP-Glo

96/384 well

E276

PKCι

ADP-Glo

96/384 well

E277

PKCμ

ADP-Glo

96/384 well

E278

PKD2

ADP-Glo

96/384 well

E279

PLK1

ADP-Glo

96/384 well

E280

PRKG1

ADP-Glo

96/384 well

E281

PYK2

ADP-Glo

96/384 well

E282

RET

ADP-Glo

96/384 well

E283

RET(V804L)

ADP-Glo

96/384 well

E284

RET(Y791F)

ADP-Glo

96/384 well

E285

RIPK2

ADP-Glo

96/384 well

E286

ROCK1

ADP-Glo

96/384 well

E287

ROCK2

ADP-Glo

96/384 well

E288

RON

ADP-Glo

96/384 well

E289

RSK1

ADP-Glo

96/384 well

E290

SGK1

ADP-Glo

96/384 well

E291

SIK

ADP-Glo

96/384 well

E292

SLK

ADP-Glo

96/384 well

E293

SRC

ADP-Glo

96/384 well

E294

STK33

ADP-Glo

96/384 well

E295

SYK

ADP-Glo

96/384 well

E296

TAK1-TAB1

ADP-Glo

96/384 well

E297

TAOK1

ADP-Glo

96/384 well

E298

TBK1

ADP-Glo

96/384 well

E299

TGFbR1

ADP-Glo

96/384 well

E300

TGFβR2

ADP-Glo

96/384 well

E301

TNIK

ADP-Glo

96/384 well

E302

TOPK

ADP-Glo

96/384 well